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Mirogabalin besylate

CAS No.: 1138245-21-2      Formula: C18H25NO5S

Weight: 367.46000

Synonyms: DS-5565 besylate; [(1R,5S,6S)-6-(aminomethyl)-3-ethylbicyclo[3.2.0]hept-3-en-6-yl]acetic acid benzenesulfonate; [(1R,5S,6S)-6-(Aminomethyl)-3-ethylbicyclo[3.2.0]hept-3-en-6-yl]acetic acid monobenzenesulfonate;


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Description

Mirogabalin (DS-5565) is a drug developed by Daiichi Sankyo and related to drugs such as gabapentin and pregabalin. Similarly to these drugs, mirogabalin binds to the α2δ calcium channels (1 and 2), but with significantly higher potency than pregabalin. It has shown promising results in Phase II clinical trials for the treatment of diabetic peripheral neuropathic pain, and is currently in Phase III trials.

Basic Information
CAS No.:
1138245-21-2
Synonyms:
DS-5565 besylate; [(1R,5S,6S)-6-(aminomethyl)-3-ethylbicyclo[3.2.0]hept-3-en-6-yl]acetic acid benzenesulfonate; [(1R,5S,6S)-6-(Aminomethyl)-3-ethylbicyclo[3.2.0]hept-3-en-6-yl]acetic acid monobenzenesulfonate;
Formula:
C18H25NO5S
Molecular Weight:
367.46000
PSA:
126.07000
LogP:
4.49680
Properties
Appearance & Character:
Density:
Melting Point:
Boiling Point:
Flash Point:
Storage Conditions:
Safety Info